Peer-Reviewed Journal Details
Mandatory Fields
Maguire, AR;Kelleher, LL;Ferguson, G
1996
June
Journal of Molecular Catalysis B: Enzymatic
Efficient kinetic resolution of 2-benzenesulfonylcyclopentanone derivatives
Validated
WOS: 12 ()
Optional Fields
DESS-MARTIN PERIODINANE BAKERS-YEAST REDUCTION MICROBIAL REDUCTION KETO ESTER SULFONES CHEMISTRY CONFIGURATION OXIDATION SULFIDES LACTONES
1
115
126
Efficient kinetic resolution of 2-benzenesulfonylcyclopentanones 1, bearing 3-alkyl, 3-aryl, or 3-benzyl substituents, has been achieved by bakers' yeast mediated reduction. With the unsubstituted 2-benzenesulfonylcyclopentanone 1a, efficient asymmetric reduction to form (1S,2R)-cis-2-benzenesulfonylcyclopentanol 2a is observed under the same conditions. Excellent enantioselectivities (up to > 95% eel are obtained.
AMSTERDAM
1381-1177
Grant Details