Peer-Reviewed Journal Details
Mandatory Fields
Mccaw, PG;Deadman, BJ;Maguire, AR;Collins, SG
2016
September
Journal of Flow Chemistry
Delivering Enhanced Efficiency in the Synthesis of alpha-Diazosulfoxides by Exploiting the Process Control Enabled in Flow
Validated
Optional Fields
MULTISTEP ORGANIC-SYNTHESIS BETA-OXO SULFOXIDES SULFINE CHEMISTRY DIAZO-COMPOUNDS TECHNOLOGY GENERATION PRODUCTS REACTORS AZIDE
6
226
233
Continuous-flow generation of alpha-diazosulfoxides results in a two- to three-fold increase in yields and decreased reaction times compared to standard batch synthesis methods. These high yielding reactions are enabled by flowing through a bed of polystyrene-supported base (PS-DBU or PS-NMe2) with highly controlled residence times. This engineered solution allows the alpha-diazosulfoxides to be rapidly synthesized while limiting exposure of the products to basic reaction conditions, which have been found to cause rapid decomposition. In addition to improved yields, this work has the added advantage of ease of processing, increased safety profile, and scale-up potential.
BUDAPEST
2062-249X
10.1556/1846.2016.00013
Grant Details